发明名称 Bicyclic amine derivatives
摘要 The invention provides a compound of formula (I):wherein A represents a bidentate group of formula -CH2-X-CH2- (wherein X is methylene, sulfur or oxygen), X'C=CY or X'WC-CYZ (wherein X', W, Y and Z are independently hydrogen, hydroxy, acyloxy, alkoxy, alkylsilyloxy, cyano or halogen, or X' and W or Y and Z together with the carbon to which they are attached form a carbonyl group), provided that A is not CH2-CH2; Ar is an optionally substituted phenyl or 5- or 6-membered heterocyclic ring system containing from 1 to 3 heteroatoms individually selected from nitrogen, oxygen and sulfur atoms, and at least one unsaturation (double bond) between adjacent atoms in the ring, said heterocyclic ring being optionally fused to a benzene ring; aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkanyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl, dithiocarboxyl moieties of R, R3 and R4 comprise from 1 to 15 carbon atoms, and are optionally substituted with one or more substituents selected from, halogen, cyano, carboxyl, carboxylic acyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxy, nitro, haloalkyl, alkyl, amino, acylamino, imidate and phosphonato groups; or an acid addition salt, quaternary ammonium salt or N-oxide derived therefrom; an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor; a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.
申请公布号 US6177442(B1) 申请公布日期 2001.01.23
申请号 US19990357750 申请日期 1999.07.21
申请人 ZENECA LIMITED 发明人 URCH CHRISTOPHER JOHN;LEWIS TERENCE;SUNLEY RAYMOND LEO;SALMON ROGER;GODFREY CHRISTOPHER RICHARD AYLES;BRIGHTWELL CHRISTOPHER IAN;HOTSON MATTHEW BRIAN
分类号 A01N43/90;A01N47/16;A01N47/18;A61K31/435;A61K31/46;A61K31/496;A61K31/5377;C07D413/14;C07D417/14;C07D451/02;C07D451/04;C07D451/06;C07D451/14;C07D471/08;C07D498/08;C07D513/08;(IPC1-7):A61K31/46 主分类号 A01N43/90
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