发明名称 Heteroaryl piperidines, heteroaryl pyrrolidines and heteroaryl piperazines, pharmaceutical preparations in which they are comprised as well as their use
摘要 <p>In the present invention there are disclosed heteroaryl piperidines, heteroaryl pyrrolidines and heteroaryl piperazines of the general formula I, in which X represents oxygen, sulfur or an optionally substituted imino group, p is a number of 1 or 2, Y represents hydrogen, a lower alkyl or alkoxyl, hydroxyl, chlorine, fluorine, bromine or iodine, trifluoromethyl, a nitro group or an amino group and Qi1 represents an organic substituent. The aforementioned compounds are effective particularly as antipsychotics and analgesics and they can be therefore used for treating psychoses and relief of pain, particularly in the form of pharmaceutical preparations.</p>
申请公布号 CZ287611(B6) 申请公布日期 2001.01.17
申请号 CZ19940001102 申请日期 1992.11.04
申请人 AVENTIS PHARMACEUTICALS INC. 发明人 STRUPCZEWSKI JOSEPH T.;HELSLEY GROVER C.;CHIANG YULIN;BORDEAU KENNETH J.;GLAMKOWSKI EDWARD J.
分类号 A61K31/09;A61K31/00;A61K31/12;A61K31/40;A61K31/41;A61K31/415;A61K31/4162;A61K31/42;A61K31/423;A61K31/425;A61K31/428;A61K31/44;A61K31/4427;A61K31/445;A61K31/4465;A61K31/4523;A61K31/454;A61K31/495;A61K31/496;A61K31/505;A61K31/506;A61K31/535;A61K31/5375;A61K31/5377;A61K31/55;A61P25/04;A61P25/18;A61P29/00;C07C45/45;C07C45/67;C07C45/71;C07C47/277;C07C47/575;C07C49/84;C07C233/25;C07C233/33;C07C255/54;C07C323/22;C07D;C07D207/08;C07D221/04;C07D231/56;C07D239/02;C07D261/20;C07D275/04;C07D275/06;C07D277/82;C07D401/04;C07D401/12;C07D401/14;C07D403/04;C07D403/12;C07D403/14;C07D405/04;C07D405/14;C07D409/14;C07D413/04;C07D413/12;C07D413/14;C07D417/04;C07D417/12;C07D417/14;C07D419/04;C07D471/04;C07F7/18;(IPC1-7):C07D261/20 主分类号 A61K31/09
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