发明名称 PROCESS FOR THE SYNTHESIS OF HIV PROTEASE INHIBITORS
摘要 <p>An improved process for the synthesis of (3S)-tetrahydro-3-furyl N-[(1S,2R)-3 -(4-amino-N-isobutylbenzenesulphonamido)-1-benzyl-2-hydroxypropyl]carbamate comprising four steps form the compound of formula A and a novel intermediate thereto.</p>
申请公布号 EP1066276(A1) 申请公布日期 2001.01.10
申请号 EP19990910543 申请日期 1999.03.18
申请人 GLAXO GROUP LIMITED 发明人 AL-FARHAN, EMILE;DEININGER, DAVID, D.;MCGHIE, STEPHEN;O'CALLAGHAN, JOHN;ROBERTSON, MARK, STUART;RODGERS, KEITH;ROUT, STEPHEN, JOHN;SINGH, HARDEV;TUNG, ROGER, DENNIS
分类号 A61P31/18;C07C311/18;C07D307/20;(IPC1-7):C07D307/20 主分类号 A61P31/18
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