发明名称 CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY
摘要 The present invention is directed to compounds of formula (I) wherein R<1>, R<2>, R<3>, R<4>, R<5>, R<7>, R<8>, X, n, x and y are defined herein which are useful as modulators of chemokine receptor activity. In particular, these compounds are useful as modulators of the chemokine receptors CCR-5 and/or CCR-3.
申请公布号 WO0076514(A1) 申请公布日期 2000.12.21
申请号 WO2000US15769 申请日期 2000.06.08
申请人 MERCK & CO., INC.;FINKE, PAUL, E.;HILFIKER, KERRY, A.;LOEBACH, JENNIFER, L.;MACCOSS, MALCOLM;MILLS, SANDER, G.;SHEN, DONG-MING;OATES, BRYAN 发明人 FINKE, PAUL, E.;HILFIKER, KERRY, A.;LOEBACH, JENNIFER, L.;MACCOSS, MALCOLM;MILLS, SANDER, G.;SHEN, DONG-MING;OATES, BRYAN
分类号 C07D211/14;C07D211/18;C07D211/24;C07D211/34;C07D401/04;C07D401/06;C07D401/12;C07D413/06;C07D417/04;C07D471/04 主分类号 C07D211/14
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