发明名称 N-CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY
摘要 <p>The present invention is directed to compounds of formula (I) (wherein R<1>, R<3>, R<4>, R<5>, R<6>, R<7>, R<8>, X, n, x and y are defined herein) which are useful as modulators of chemokine receptor activity. In particular, these compounds are useful as modulators of the chemokine receptors CCR-5 and/or CCR-3.</p>
申请公布号 WO0076972(A1) 申请公布日期 2000.12.21
申请号 WO2000US15736 申请日期 2000.06.08
申请人 MERCK & CO., INC.;FINKE, PAUL, E.;HILFIKER, KERRY, A.;MACCOSS, MALCOLM;CHAPMAN, KEVIN, T.;LOEBACH, JENNIFER, L.;MILLS, SANDER, G.;GUTHIKONDA, RAVI, N.;SHAH, SHRENIK, K.;KIM, DOOSEOP;SHEN, DONG-MING;OATES, BRYAN 发明人 FINKE, PAUL, E.;HILFIKER, KERRY, A.;MACCOSS, MALCOLM;CHAPMAN, KEVIN, T.;LOEBACH, JENNIFER, L.;MILLS, SANDER, G.;GUTHIKONDA, RAVI, N.;SHAH, SHRENIK, K.;KIM, DOOSEOP;SHEN, DONG-MING;OATES, BRYAN
分类号 C07D487/04;A61K31/437;A61K31/445;A61K31/4468;A61K31/4525;A61K31/454;A61K31/4545;A61K31/4709;A61K31/506;A61P9/10;A61P11/02;A61P11/06;A61P17/00;A61P19/02;A61P27/02;A61P29/00;A61P31/00;A61P31/18;A61P37/00;A61P37/02;A61P37/08;A61P43/00;C07D211/14;C07D211/18;C07D211/20;C07D211/24;C07D211/30;C07D211/34;C07D211/58;C07D277/30;C07D401/04;C07D401/06;C07D401/12;C07D401/14;C07D405/14;C07D413/04;C07D413/06;C07D417/04;C07D471/04;(IPC1-7):C07D211/14;A61K31/440;C07D263/32;C07D231/12;C07D239/42;C07D271/12 主分类号 C07D487/04
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