发明名称 |
INDOLYLPIPERIDINE DERIVATIVES AS ANTIHISTAMINIC AND ANTIALLERGIC AGENTS |
摘要 |
Indolylpiperidine compounds of formula (I) wherein: A1 represents an alkylen e, alkyleneoxy, alkylenethio, alkanoyl or hydroxyalkylene group; A2 represents a single bond, an alkylene or alkenylene group; W represents a single bond or a phenylene or furanylene group which is unsubstituted or substituted by one o r more halogen atoms, alkoxy groups and/or alkyl groups; R2 represents a hydrogen or halogen atom or an alkyl or alkoxy group; and R3 represents a carboxyl group or a tetrazolyl group. The present invention provides novel indolylpiperidine compounds having improved antihistamine and antiallergic activity.
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申请公布号 |
CA2375985(A1) |
申请公布日期 |
2000.12.14 |
申请号 |
CA20002375985 |
申请日期 |
2000.05.31 |
申请人 |
ALMIRALL PRODESFARMA S.A. |
发明人 |
FERNANDEZ FORNER, DOLORS;PAGES SANTACANA, LLUIS;FONQUERNA POU, SILVIA;PUIG DURAN, CARLES |
分类号 |
A61K31/445;A61K31/4525;A61K31/454;A61P11/02;A61P11/04;A61P11/06;A61P27/02;A61P37/08;C07D401/04;C07D401/14;C07D405/14;(IPC1-7):C07D401/04 |
主分类号 |
A61K31/445 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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