发明名称 Novel catechols as antimicrobial agents
摘要 Compounds, pharmaceutically acceptable salts, and compositions thereof of the general formula:wherein Ar is aryl and heteroaryl; R1, R2, R3, and R4 are hydrido, alkyl, cyano, heteroaryl, hydroxy, amino, acylamino, halo, alkoxy, aryloxy, carboxyamido, alkenyl, cycloalkyl, heterocyclyl, acyl, acyloxy, carboalkoxy, carboxy, thio, sulfinyl, sulfonyl and sulfoxy, R5, R6, R7, and R8 are hydrido and lower alkyl; and Het is a nitrogen-containing heterocyclic ring.
申请公布号 AU4819900(A) 申请公布日期 2000.11.17
申请号 AU20000048199 申请日期 2000.05.05
申请人 MERCK & CO., INC.;CUBIST PHARMACEUTICALS, INC. 发明人 AARON H. LEEMAN;MILTON L. HAMMOND;MILANA MALETIC;GINA M. SANTORELLI;SHERMAN F. WADDELL;JOHN FINN;MICHAEL MORYTKO;JASON HILL;DENNIS KEITH
分类号 A61K31/4184;A61K31/437;A61K31/454;A61P31/04;A61P31/10;C07D215/14;C07D233/54;C07D235/12;C07D401/12;C07D403/12;C07D405/12;C07D471/04;C07D521/00 主分类号 A61K31/4184
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