发明名称 |
PROSES UNTUK SINTESA ANALOG-ANALOG NUKLEOSIDA |
摘要 |
<p>The present invention relates to an improved method for synthesizing nucleosides with a low alpha : beta anomeric ratio. The method comprises coupling a protected furanosyl halide and an appropriately protected heterocycle in the presence of a nucleophilic polar solvent and a strong base.</p> |
申请公布号 |
ID25992(A) |
申请公布日期 |
2000.11.16 |
申请号 |
ID20000000389D |
申请日期 |
2000.05.10 |
申请人 |
PFIZER PRODUCTS INC. |
发明人 |
ROBERT WILLIAM SCOTT |
分类号 |
C07H19/14;B01J31/02;C07B61/00;C07H19/04;C07H19/06;C07H19/16;C07H19/23;C07H21/00;(IPC1-7):C07D411/04 |
主分类号 |
C07H19/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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