发明名称 |
RINGSUBSTITUIERTE 2-AMINO-1,2,3,4- TETRAHYDRONAPHTAHLINE UND 3-AMINOCHROMANE |
摘要 |
<p>Isoxazole derivs. of formula (I) and their acid-addn. salts and solvates are new: In (I) R = 1-4C alkyl, allyl or cyclopropylmethyl; R1 = H, 1-4C alkyl, allyl, cyclopropylmethyl or aryl(1-4C)alkyl; X = CH2 or O; y = 4-R2-5-R3-3-isoxazolyl or 3-R2-4-R3-5-isoxazolyl; R2 and R3 = H, 1-4C alkyl, 1-4C alkoxy, 1-4C alkylthio, OH, NH2, CN or Ph. Pref. x = CH2; R and R1 = 1-4C alkyl, esp. n-Pr; R2 and R3 = H.</p> |
申请公布号 |
AT197145(T) |
申请公布日期 |
2000.11.15 |
申请号 |
AT19960200393T |
申请日期 |
1992.02.03 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
HOECHSTETTER, CRAIG S.;HUSER, DIANE L.;SCHAUS, JOHN M.;TITUS, ROBERT D. |
分类号 |
A61K31/42;A61K31/353;A61K31/4015;A61P1/00;A61P1/14;A61P9/12;A61P13/02;A61P15/00;A61P25/00;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/26;A61P25/32;A61P43/00;C07C225/18;C07C225/20;C07C255/42;C07C323/29;C07D261/08;C07D261/10;C07D261/12;C07D261/14;C07D261/18;C07D311/04;C07D311/20;C07D311/58;C07D413/04;C07D413/10;(IPC1-7):C07C225/20;C07C211/42 |
主分类号 |
A61K31/42 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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