发明名称 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN
摘要 Novel boronic acid and ester and carboxyl-modified amino acid compounds of the Formula I, which are inhibitors of trypsin-like enzymes, are disclosed:R1-Z-CHR2-A,where R1, Z, R2 and A are defined within.
申请公布号 EP0810858(A4) 申请公布日期 2000.11.15
申请号 EP19950944331 申请日期 1995.12.13
申请人 DUPONT PHARMACEUTICALS COMPANY 发明人 AMPARO, EUGENE CRUZ;MILLER, WILLIAM HENRY;PACOFSKY, GREGORY JAMES;WITYAK, JOHN;WEBER, PATRICIA CAROL;DUNCIA, JOHN JONAS VYTAUTAS;SANTELLA, JOSEPH BASIL, III
分类号 C07D249/08;C07F5/02 主分类号 C07D249/08
代理机构 代理人
主权项
地址