发明名称 SUBSTITUTED 2-ARYLIMINO HETEROCYCLES AND COMPOSITIONS CONTAINING THEM, FOR USE AS PROGESTERONE RECEPTOR BINDING AGENTS
摘要 This invention relates to 2-arylimino heterocycles, including 2-arylimino-1, 3-thiazolidines, 2-arylimino-2, 3, 4, 5-tetrahydro-1, 3-thiazines, 2-arylimino-1, 3-thiazolidin-4-ones, 2-arylimino-1, 3-thiazolidin-5-ones, and 2-arylimino-1, 3-oxazolidines, and their use in modulating progesterone receptor mediated processes, and pharmaceutical compositions for use in such therapies.
申请公布号 WO0042031(A3) 申请公布日期 2000.11.09
申请号 WO1999US29601 申请日期 1999.12.14
申请人 BAYER CORPORATION 发明人 DIXON, BRIAN, R.;BAGI, CEDO, M.;BRENNAN, CATHERINE, R.;BRITTELLI, DAVID, R.;BULLOCK, WILLIAM, H.;CHEN, JINSHAN;COLLIBEE, WILLIAM, L.;DALLY, ROBERT;JOHNSON, JEFFREY, S.;KLUENDER, HAROLD, C., E.;LATHROP, WILLIAM, F.;LIU, PEIYING;MASE, CAROL, ANN;REDMAN, ANIKO, M.;SCOTT, WILLIAM, J.;URBAHNS, KLAUS;WOLANIN, JOHN, J.
分类号 C07D233/42;A61K;A61K31/4164;A61K31/421;A61K31/423;A61K31/425;A61K31/426;A61K31/427;A61K31/428;A61K31/429;A61K31/437;A61K31/54;A61K31/55;A61P;A61P5/00;A61P5/24;A61P9/00;A61P9/10;A61P13/00;A61P15/00;A61P15/04;A61P15/08;A61P15/10;A61P15/16;A61P15/18;A61P17/00;A61P19/00;A61P19/10;A61P25/00;A61P25/24;A61P25/28;A61P35/00;A61P41/00;C07D;C07D263/28;C07D263/52;C07D277/18;C07D277/20;C07D277/42;C07D277/54;C07D277/60;C07D279/06;C07D281/02;C07D417/06;C07D417/12;C07D513/04;C07D513/10;(IPC1-7):C07D277/18 主分类号 C07D233/42
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