发明名称 Selective epoxidation process for preparing pharmaceutical compounds
摘要 PCT No. PCT/US98/03667 Sec. 371 Date Aug. 24, 1999 Sec. 102(e) Date Aug. 24, 1999 PCT Filed Feb. 25, 1998 PCT Pub. No. WO98/38164 PCT Pub. Date Sep. 3, 1998Cryptophycin compounds possessing a beta -epoxy moiety may be made with high stereoselectivity at various steps in the overall synthetic process. This invention also provides novel intermediates useful in preparing Cryptophycin compounds.
申请公布号 US6143909(A) 申请公布日期 2000.11.07
申请号 US19990380005 申请日期 1999.08.24
申请人 ELI LILLY AND COMPANY 发明人 HOARD, DAVID WARREN;MOHER, ERIC DAVID;PATEL, VINOD FRANCIS;NORMAN, BRYAN HURST
分类号 C07D303/38;C07D303/40;C07D303/46;C07D405/06;C07D405/12;C07D413/06;(IPC1-7):C07D303/38;C07D301/02 主分类号 C07D303/38
代理机构 代理人
主权项
地址