发明名称 |
Selective epoxidation process for preparing pharmaceutical compounds |
摘要 |
PCT No. PCT/US98/03667 Sec. 371 Date Aug. 24, 1999 Sec. 102(e) Date Aug. 24, 1999 PCT Filed Feb. 25, 1998 PCT Pub. No. WO98/38164 PCT Pub. Date Sep. 3, 1998Cryptophycin compounds possessing a beta -epoxy moiety may be made with high stereoselectivity at various steps in the overall synthetic process. This invention also provides novel intermediates useful in preparing Cryptophycin compounds.
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申请公布号 |
US6143909(A) |
申请公布日期 |
2000.11.07 |
申请号 |
US19990380005 |
申请日期 |
1999.08.24 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
HOARD, DAVID WARREN;MOHER, ERIC DAVID;PATEL, VINOD FRANCIS;NORMAN, BRYAN HURST |
分类号 |
C07D303/38;C07D303/40;C07D303/46;C07D405/06;C07D405/12;C07D413/06;(IPC1-7):C07D303/38;C07D301/02 |
主分类号 |
C07D303/38 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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