发明名称 |
Preparation of [1S-[1A,2B,3B,4A(S*)]]-4-[7-[[1-(3-chloro-2-thienyl)methyl propyl]amino]-3H-imidazo[4,5-B]pyridin-3-yl]-N-ethyl-2,3-dihydroxycyclopentanecarboxamide |
摘要 |
This invention is directed to methods for the preparation of [1S-[1a,2b,3b,4a(S*)]]-4-[7-[[1-(3-chloro-2-thienyl) methyl]propyl]amino]-3H-imidazo[4,5-b]pyridin-3-yl]-N-ethyl-2,3-dihydroxycyclopentanecarboxamide, methods for the preparation of intermediates thereto, and to said intermediates themselves.
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申请公布号 |
US6143894(A) |
申请公布日期 |
2000.11.07 |
申请号 |
US19990233591 |
申请日期 |
1999.01.19 |
申请人 |
AVENTIS PHARMACEUTICALS PRODUCTS INC. |
发明人 |
O'BRIEN, MICHAEL K.;GARCIA, HERVE;LEON, PATRICK;POWNER, TORY H.;REILLY, LAURENCE W.;SHAH, HARSHAVADAN C.;THOMPSON, MICHAEL D.;TSUEI, CHING T.;VANASSE, BENOIT J.;WALTHER, FRANCIS L. |
分类号 |
A61P3/06;A61P9/00;A61P9/12;C07D213/69;C07D409/12;C07D409/14;C07D471/04;(IPC1-7):C07D471/04 |
主分类号 |
A61P3/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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