| 发明名称 |
Taxoid compound and method for producing the same |
| 摘要 |
A taxoid compound represented by general formula (I) where the symbols R1, R2, R3, R4, Bz, and Ac have specified meanings. Also, a method for producing the taxoid derivative from a baccatin derivative having a beta -ketoester group at the 13-position by transesterification and a method for producing taxoid compound such as paclitaxel from the taxoid derivative under mild condition are disclosed.
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| 申请公布号 |
US6136990(A) |
申请公布日期 |
2000.10.24 |
| 申请号 |
US20000504788 |
申请日期 |
2000.02.15 |
| 申请人 |
BIO RESEARCH CORPORATION OF YOKOHAMA;ENSUIKO SUGAR REFINING CO., LTD.;MANDAI, TADAKATSU |
发明人 |
MANDAI, TADAKATSU;OKUMOTO, HIROSHI;NAKANISHI, KATSUYOSHI;HARA, KOJI;MIKUNI, KATSUHIKO;HARA, KOZO |
| 分类号 |
C07D305/14;C07D413/12;(IPC1-7):C07D305/14;C07D409/00;C07D405/00 |
主分类号 |
C07D305/14 |
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