发明名称 PREPARATION OF [1S-[1A,2B,3B,4A(S*)]]-4-[7-[[1-(3-CHLORO-2-THIENYL) METHYL]PROPYL]AMINO]-3H-IMIDAZO[4,5-B]PYRIDIN-3-YL]-N-ETHYL-2,3-DIHYDROXYCYCLOPENTANECARBOXAMIDE
摘要 This invention is directed to methods for the preparation of ¢1S¢1a,2b,3b,4a(S*)!!-4-¢7-¢¢1-(3-chloro-2-thienyl)methyl!propyl!amino!-3H-imidazo¢4,5-b!pyridin-3-yl!-N-ethyl-2,3-dihydroxycyclopentanecarboxamide, methods for the preparation of intermediates thereto, and to said intermediates themselves.
申请公布号 CA2274630(C) 申请公布日期 2000.10.03
申请号 CA19972274630 申请日期 1997.11.24
申请人 RHONE-POULENC RORER PHARMACEUTICALS INC. 发明人 LEON, PATRICK;REILLY, LAURENCE W.;GARCIA, HERVE;SHAH, HARSHAVADAN C.;VANASSE, BENOIT J.;TSUEI, CHING T.;POWNER, TORY H.;THOMPSON, MICHAEL D.;WALTHER, FRANCIS L.;O'BRIEN, MICHAEL K.
分类号 A61P3/06;A61P9/00;A61P9/12;C07D213/69;C07D409/12;C07D409/14;C07D471/04;(IPC1-7):C07D409/12 主分类号 A61P3/06
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