发明名称 |
Method for making cocaine receptor binding ligands and intermediates therefor |
摘要 |
An improved method for preparation of cocaine receptor binding ligands is provided. The method calls for the preparation of the silylaryl intermediate prepared from phenyl trimethylsilane and a anhydroecgonine methyl ester appropriately substituted. The intermediate is prepared in high purity and can be directly converted to the binding ligand by iodine substitution.
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申请公布号 |
US6123917(A) |
申请公布日期 |
2000.09.26 |
申请号 |
US19950509055 |
申请日期 |
1995.07.31 |
申请人 |
RESEARCH TRIANGLE INSTITUTE |
发明人 |
CARROLL, FRANK IVY |
分类号 |
A61K51/04;C07D451/02;C07F7/08;C07F7/22;(IPC1-7):A61K51/04;C07D401/00 |
主分类号 |
A61K51/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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