发明名称 Crystal modification d of 8-cyano-1-cyclopropyl-7- (1s, 6s- 2,8- diazabicyclo- (4.3.0) nonan-8-yl) -6-fluoro -1,4-dihydro -4-oxo -3-quinoline carboxylic acid
摘要 The present invention relates to a defined crystal modification of 8-cyano-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo[4.3.0]nonan-8-yl)-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid, to processes for its preparation and to its use in pharmaceutical preparations.The crystal modification can be distinguished from other crystal modifications of 8-cyano-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo[4.3.0]nonan-8-yl)-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid of the formula (I) by its characteristic X-ray powder diffractogram and its differential thermodiagram (see description).
申请公布号 AU3154400(A) 申请公布日期 2000.09.21
申请号 AU20000031544 申请日期 2000.02.14
申请人 BAYER AKTIENGESELLSCHAFT 发明人 THOMAS HIMMLER;HUBERT RAST
分类号 A61K31/4709;A61P31/04;C07D471/04 主分类号 A61K31/4709
代理机构 代理人
主权项
地址