发明名称 |
Dihydrochloride pseudo-polymorphous forms of 2-[2-[4-[bis(4-fluorophenyl)methyl]-1-piperazinyl]ethoxy]acetic acid |
摘要 |
<p>The present invention relates to new pseudopolymorphic forms of 2-Ä2-Ä4-Äbis(4-fluorophenyl)methylÜ-1-piperazinylÜethoxyÜacetic acid dihydrochloride, namely, anhydrous 2-Ä2-Ä4-Äbis(4-fluorophenyl)methylÜ-1-piperazinylÜethoxyÜacetic acid dihydrochloride and 2-Ä2-Ä4-Äbis(4-fluorophenyl)methylÜ-1-piperazinylÜethoxyÜacetic acid dihydrochloride monohydrate. It also relates to processes for the preparation of these pseudopolymorphic forms and to pharmaceutical compositions containing them.</p> |
申请公布号 |
CZ20001787(A3) |
申请公布日期 |
2000.09.13 |
申请号 |
CZ20000001787 |
申请日期 |
1998.11.26 |
申请人 |
UCB, S. A. |
发明人 |
BERWAER MONIQUE;BODSON GUY;DELEERS MICHEL;DOGIMONT CHARLES;FANARA DOMENICO;TIMMERMANS JACQUES |
分类号 |
C07D295/08;A61K31/495;A61P11/08;A61P17/00;A61P25/08;A61P37/08;A61P43/00;C07D295/084;C07D295/088;(IPC1-7):C07D295/08 |
主分类号 |
C07D295/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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