| 发明名称 |
Process for preparing protease inhibitor |
| 摘要 |
<p>Disclosed is a novel process and novel intermediates to prepare [R-(R*,R*)]-N-[3-[1-[5,6-dihydro-4-hydroxy-2-oxo-6-(2-phenylethyl)-6-propyl-2H-pyran-3-yl]propyl]phenyl]-5-(trifluoromethyl)-2-pyridinesulfonamide (XIX) which is a protease inhibitor useful in treating humans infected with the HIV virus.</p> |
| 申请公布号 |
CZ20000804(A3) |
申请公布日期 |
2000.08.16 |
| 申请号 |
CZ20000000804 |
申请日期 |
1998.09.03 |
| 申请人 |
PHARMACIA & UPJOHN COMPANY |
发明人 |
GAGE JAMES R.;KELLY ROBERT C.;HEWITT BRADLEY D. |
| 分类号 |
C07C205/43;A61K31/366;A61P31/18;C07C45/30;C07C47/277;C07C59/48;C07C201/16;C07C205/56;C07D309/32;C07D405/04;C07D405/12;(IPC1-7):C07D309/32 |
主分类号 |
C07C205/43 |
| 代理机构 |
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