发明名称 |
Benzoheterocyclic derivatives |
摘要 |
PCT No. PCT/JP95/01124 Sec. 371 Date Nov. 13, 1996 Sec. 102(e) Date Nov. 13, 1996 PCT Filed Jun. 7, 1995 PCT Pub. No. WO95/34540 PCT Pub. Date Dec. 21, 1995A benzoheterocyclic derivative of the following formula [1]: and pharmaceutically acceptable salts thereof, which show excellent anti-vasopressin activity, vasopressin agonistic activity and oxytocin antagonistic activity, and are useful as a vasopressin antagonist, vasopressin agonist or oxytocin antagonist.
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申请公布号 |
US6096735(A) |
申请公布日期 |
2000.08.01 |
申请号 |
US19960737432 |
申请日期 |
1996.11.13 |
申请人 |
OTSUKA PHARMACEUTICAL COMPANY, LIMITED |
发明人 |
OGAWA, HIDENORI;KONDO, KAZUMI;YAMASHITA, HIROSHI;KAN, KEIZO;MATSUZAKI, TAKAYUKI;SHINOHARA, TOMOICHI;TANADA, YOSHIHISA;KURIMURA, MUNEAKI;TOMINAGA, MICHIAKI;YABUUCHI, YOICHI |
分类号 |
A61K31/55;A61K31/551;A61P1/08;A61P1/16;A61P3/10;A61P3/12;A61P5/40;A61P7/02;A61P7/04;A61P7/10;A61P9/04;A61P9/08;A61P9/10;A61P9/12;A61P13/00;A61P13/12;A61P15/04;A61P15/08;A61P15/14;A61P25/00;A61P43/00;C07D215/12;C07D215/18;C07D223/16;C07D243/12;C07D243/14;C07D401/06;C07D401/10;C07D401/12;C07D401/14;C07D403/06;C07D403/10;C07D403/12;C07D405/12;C07D409/06;C07D413/10;C07D417/06;C07D417/10;C07D471/04;C07D521/00;(IPC1-7):C07D223/16;A61K31/47 |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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