发明名称 THIAZOLE DERIVATIVES AS PPAR GAMMA LIGANDS
摘要 The present invention discloses novel PPARgamma ligands of Formula (I) and pharmaceutically acceptable salts and solvates thereof. The present invention also discloses a method for treating osteoporosis by administration of a PPARgamma antagonist. n=2 - 4 and R1 - R5 are as in the application.
申请公布号 WO0027832(A3) 申请公布日期 2000.07.27
申请号 WO1999EP08477 申请日期 1999.11.09
申请人 GLAXO GROUP LIMITED;COLLINS, JON, LOREN;HOLMES, CHRISTOPHER, PATRICK;LENHARD, JAMES, MARTIN;WILLSON, TIMOTHY, MARK 发明人 COLLINS, JON, LOREN;HOLMES, CHRISTOPHER, PATRICK;LENHARD, JAMES, MARTIN;WILLSON, TIMOTHY, MARK
分类号 A61K31/425;A61K31/426;A61K31/427;A61K31/443;A61K31/4439;A61P3/00;A61P3/04;A61P3/10;A61P9/00;A61P19/10;A61P29/00;A61P35/00;A61P43/00;C07D277/14;C07D417/06;C07D417/10;C07D417/12;G01N33/566 主分类号 A61K31/425
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