| 发明名称 |
METHOD FOR PREPARING AN AZA-MACROLIDE WITH 4'' (R) NH2 |
| 摘要 |
The invention concerns a method for regioselective preparation of a compound of general formula (I) by regioselective displacement with a nitrogenous nucleophile of the activated alcohol function in position 4'' of a corresponding derivative of general formula (II).
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| 申请公布号 |
WO0042056(A1) |
申请公布日期 |
2000.07.20 |
| 申请号 |
WO2000FR00089 |
申请日期 |
2000.01.17 |
| 申请人 |
MERIAL |
发明人 |
LEON, PATRICK;LHERMITTE, FREDERIC;GUEVEL, RONAN;PAUZE, DENIS;GAREL, LAURENT;ODDON, GILLES |
| 分类号 |
A61K31/70;A61P31/00;C07B61/00;C07H17/08;(IPC1-7):C07H17/08 |
主分类号 |
A61K31/70 |
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