摘要 |
Novel compounds exhibiting chymase-inhibiting activities and being useful as various drugs, i.e., SF2809-I, SF2809-II, SF2809-III, SF2809-IV, SF2809-V and SF2809-VI substances represented by general formula (VII), and pharmaceutically acceptable salts thereof: [wherein R<1> is hydrogen, phenyl or p-hydroxyphenyl; and R<2> is acetylamino(-NHCOCH3) or hydroxyl]; a process for the preparation of SF2809 substances; and drug compositions containing the same.
|
申请人 |
MEIJI SEIKA KAISHA, LTD.;TEIJIN LTD.;TANI, MASATO;GYOBU, YASUHIRO;MORIYAMA, CHIEKO;SASAKI, TORU;TAKENOUCHI, OSAMI;KAWAMURA, TAKASHI;KAMIMURA, TAKASHI;HARADA, TOSHIAKI |
发明人 |
TANI, MASATO;GYOBU, YASUHIRO;MORIYAMA, CHIEKO;SASAKI, TORU;TAKENOUCHI, OSAMI;KAWAMURA, TAKASHI;KAMIMURA, TAKASHI;HARADA, TOSHIAKI |