发明名称 SF2809-I, II, III, IV, V AND VI SUBSTANCES EXHIBITING CHYMASE-INHIBITING ACTIVITIES
摘要 Novel compounds exhibiting chymase-inhibiting activities and being useful as various drugs, i.e., SF2809-I, SF2809-II, SF2809-III, SF2809-IV, SF2809-V and SF2809-VI substances represented by general formula (VII), and pharmaceutically acceptable salts thereof: [wherein R<1> is hydrogen, phenyl or p-hydroxyphenyl; and R<2> is acetylamino(-NHCOCH3) or hydroxyl]; a process for the preparation of SF2809 substances; and drug compositions containing the same.
申请公布号 WO0032587(A1) 申请公布日期 2000.06.08
申请号 WO1999JP06738 申请日期 1999.12.01
申请人 MEIJI SEIKA KAISHA, LTD.;TEIJIN LTD.;TANI, MASATO;GYOBU, YASUHIRO;MORIYAMA, CHIEKO;SASAKI, TORU;TAKENOUCHI, OSAMI;KAWAMURA, TAKASHI;KAMIMURA, TAKASHI;HARADA, TOSHIAKI 发明人 TANI, MASATO;GYOBU, YASUHIRO;MORIYAMA, CHIEKO;SASAKI, TORU;TAKENOUCHI, OSAMI;KAWAMURA, TAKASHI;KAMIMURA, TAKASHI;HARADA, TOSHIAKI
分类号 A61P9/00;A61P11/00;A61P11/06;A61P13/12;A61P17/00;A61P27/14;A61P29/00;A61P43/00;C07D401/06;(IPC1-7):C07D401/06;C12P17/16;A61K31/470;C12N9/99 主分类号 A61P9/00
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