发明名称 Crystal form of N-(4-trifluoromethylphenyl)-5-methylisoxazole-4-carboxamide
摘要 The invention relates to a crystal modification of the compound of the formula I and the processes for the preparation of and use that crystal modifications 1. The invention is used for treating acute immunological episodes, such as sepsis, allergies, graft-versus-host and host-versus-graft-reactions, autoimmune diseases, in particular rheumatoid arthritis, systemic lupus erythematosus, multiple sclerosis, psoriasis, atopic dermatitis, asthma, urticaria, rhinitis, uveitis, type II diabetes, liver fibrosis, cystic fibrosis, colitis, cancers, such as lung cancer, leukemia, ovarian cancer, sarcomas, Kaposi's sarcoma, meningioma, intestinal cancer, lymphatic cancer, brain tumors, breast cancer, pancreatic cancer, prostate cancer, or skin cancer.
申请公布号 US6060494(A) 申请公布日期 2000.05.09
申请号 US19980129783 申请日期 1998.08.06
申请人 HOECHST MARION ROUSSEL DEUTSCHLAND GMBH 发明人 FAASCH, HOLGER;HEDTMANN, UDO;WESTENFELDER, UWE;PAULUS, ERICH
分类号 A61K31/42;A61P1/00;A61P3/08;A61P11/00;A61P13/02;A61P15/00;A61P17/00;A61P25/00;A61P27/02;A61P27/14;A61P29/00;A61P31/04;A61P35/00;A61P37/00;A61P37/08;B01D9/02;C07D261/18;(IPC1-7):A61K31/42;C07D261/08 主分类号 A61K31/42
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