发明名称 |
aqueous medicaments containing 9-hydroxy-risperidone fatty acid ester |
摘要 |
A pharmaceutical composition suitable as a depot formulation for administration by intramuscular or subcutaneous injection is claimed comprises: a) as an active ingredient, a therapeutically effective amount of a 9-hydroxy-risperidone fatty acid ester of the formula (I) or a salt, stereoisomeric or stereoisomeric mixture thereof wherein R is alkyl and b) a pharmaceutically carrier; characterised in that the pharmaceutically acceptable carrier is water and the active ingredient is suspended therein.
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申请公布号 |
NZ330369(A) |
申请公布日期 |
2000.04.28 |
申请号 |
NZ19970330369 |
申请日期 |
1997.05.12 |
申请人 |
JANSSEN PHARMACEUTICA NV |
发明人 |
EMBRECHTS, ROGER CAROLUS AUGUSTA;BORGHIJS, HERMAN KAREL;MONBALIU, JOHAN;FRANCOIS, MARC KAREL JOZEF |
分类号 |
C07D471/04;A61K9/00;A61K9/10;A61K31/505;A61K31/517;A61K31/519;A61K47/00;A61K47/02;A61K47/10;A61K47/26;A61K47/38;A61P25/00;(IPC1-7):A61K31/505 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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