发明名称 SELECTIVE EPOXIDISING PROCESS FOR USE IN PRODUCTION OF PHARMACEUTIC COMPOUNDS
摘要 Cryptophycin compounds may be prepared utilizing an epoxidation step early in the synthetic process under the conditions set forth herein. This invention also relates to novel intermediates generated by this early epoxidation process.
申请公布号 PL335347(A1) 申请公布日期 2000.04.25
申请号 PL19980335347 申请日期 1998.02.25
申请人 ELI LILLY & CO.MPANY;UNIVERSITY OF HAWAII;WAYNE STATE UNIVERSITY 发明人 PATEL VINOD FRANCIS;HOARD DAVID WARREN;MOHER ERIC DAVID;NORMAN BRYAN HURST
分类号 C07D303/16;A61K31/395;A61P35/00;C07C229/08;C07C271/22;C07D233/54;C07D277/30;C07D301/03;C07D303/38;C07D303/40;C07D303/46;C07D405/06;C07D405/12;C07D413/06;C07F7/18 主分类号 C07D303/16
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