A process for safely preparing methylamine derivatives by reacting an amine with trimethyl phosphite and an oxidizing agent such as N-halogenoamide; and novel {dimethyl}{N-[3-(4-methylphenyl)-8,9-dihydro-7H-benzocycloheptenecarbonyl]-4-aminobenzyl}{4-tetrahydropyranyl}ammonium compounds.
申请公布号
WO0021916(A1)
申请公布日期
2000.04.20
申请号
WO1999JP05674
申请日期
1999.10.14
申请人
TAKEDA CHEMICAL INDUSTRIES, LTD.;IKEMOTO, TOMOMI;KAWARAZAKI, TADAO;HASHIMOTO, HIDEO;TOMIMATSU, KIMINORI;ITO, TATSUYA;NISHIGUCHI, ATSUKO