发明名称 PHOSPHONIC ACIDS DERIVATIVES AS INHIBITORS OF PTP-1B
摘要 The invention encompasses the novel class of compounds represented by formula (I) which are inhibitors of the PTP-1B enzyme. The invention also encompasses pharmaceutical compositions and methods of treating or preventing PTP-1B mediated diseases.
申请公布号 WO0017211(A1) 申请公布日期 2000.03.30
申请号 WO1999CA00864 申请日期 1999.09.21
申请人 MERCK FROSST CANADA & CO.;LEBLANC, YVES;DUFRESNE, CLAUDE;WANG, ZHAOYIN;LI, CHUN, SING;GAUTHIER, JACQUES, Y.;THERIEN, MICHEL;LAU, CHEUK, K.;ROY, PATRICK 发明人 LEBLANC, YVES;DUFRESNE, CLAUDE;WANG, ZHAOYIN;LI, CHUN, SING;GAUTHIER, JACQUES, Y.;THERIEN, MICHEL;LAU, CHEUK, K.;ROY, PATRICK
分类号 A61K45/00;A61K31/66;A61K31/662;A61K31/663;A61P3/04;A61P3/10;A61P43/00;C07F9/38;C07F9/553;C07F9/6506;C07F9/6518;C07F9/6524;C07F9/653;C07F9/6539;C07F9/6541;H04L12/56;H04M3/00;H04M3/42;H04Q3/62;(IPC1-7):C07F9/38;C07F9/651;C07F9/652;C07F9/654;C07F9/650 主分类号 A61K45/00
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