发明名称 |
Kappa agonist compounds and pharmaceutical formulations thereof |
摘要 |
Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics are provided.The compounds of formula having the structure:whereinR1, R2, and X Y, Z, Ar and n are as described in the specification. |
申请公布号 |
AU4442899(A) |
申请公布日期 |
2000.03.27 |
申请号 |
AU19990044428 |
申请日期 |
1999.06.16 |
申请人 |
ADOLOR CORPORATION |
发明人 |
WEI YUAN ZHANG;ALAN L. MAYCOCK;MICHAEL ANTHONY MARELLA;VIRENDRA KUMAR;FORREST GAUL;AN-CHIH CHANG;DEQI GUO |
分类号 |
C07D295/12;A61K31/40;A61K31/4025;A61K31/403;A61K31/404;A61K31/4402;A61K31/4427;A61K31/443;A61K31/4439;A61K31/496;A61K31/662;A61K31/675;A61K45/00;A61K45/06;A61P25/04;A61P43/00;C07D207/12;C07D209/04;C07D209/42;C07D213/40;C07D213/56;C07D241/04;C07D295/073;C07D307/52;C07D401/14;C07D403/06;C07D403/14;C07D405/14 |
主分类号 |
C07D295/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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