发明名称 Process for preparing trovafloxacin acid salts
摘要 Trovafloxacin acid salts are prepared via the hydrolysis of imine intermediates using mineral acid including, but not limited to, methanesulfonic acid, ethanesulfonic acid, benzenesulfonic acid, nitric acid, sulfuric acid, phosphoric acid, hydrochloric acid, hydrobromic acid, tartaric acid, citric acid, acetic acid, and maleic acid. Trovafloxacin acid salts are useful as antibiotic agents.
申请公布号 AU4482699(A) 申请公布日期 2000.03.16
申请号 AU19990044826 申请日期 1999.08.27
申请人 PFIZER PRODUCTS INC. 发明人 TIMOTHY NORRIS;KEITH MICHAEL DEVRIES;PETER ROBERT ROSE
分类号 C07D401/14;A61K31/4375;A61P31/04;C07D209/52;C07D471/04 主分类号 C07D401/14
代理机构 代理人
主权项
地址