发明名称 COMPOUNDS USEFUL AS AICARFT INHIBITORS
摘要 Coumpounds of the formula (I) (where R<1>, R<2>, and R<3> are as defined in the specification) are inhibitors of AICARFT. These compounds, as well as their pharmaceutically acceptable salts, solvates, prodrugs, and pharmaceutically active metabolites, are useful in pharmaceutical compositions for treating diseases such as cancer.
申请公布号 WO0013688(A1) 申请公布日期 2000.03.16
申请号 WO1999US20331 申请日期 1999.09.03
申请人 AGOURON PHARMACEUTICALS, INC.;BLECKMAN, TED, MICHAEL;PALMER, CYNTHIA, LOUISE;ROMINES, WILLIAM, HENRY, III;VARNEY, MICHAEL, DAVID 发明人 BLECKMAN, TED, MICHAEL;PALMER, CYNTHIA, LOUISE;ROMINES, WILLIAM, HENRY, III;VARNEY, MICHAEL, DAVID
分类号 C07D409/12;C07D409/14;(IPC1-7):A61K31/505;A61K31/535;C07D239/02;C07D413/02;C07D413/14 主分类号 C07D409/12
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