发明名称 FORMAMIDE COMPOUNDS AS THERAPEUTIC AGENTS
摘要 A family of compounds having general structural formula (I) where W is a reverse hydroxamic acid group, and R1, R2, R3, R4, R5 and R6 are as described in the specification, or a pharmaceutically acceptable salt, solvate, biohydrolyzable ester, biohydrolyzable amide, affinity reagent, or prodrug thereof. Also described are methods for their preparation, pharmaceutical compositions including such compounds and their use in medicine.
申请公布号 WO0012082(A1) 申请公布日期 2000.03.09
申请号 WO1999US18960 申请日期 1999.08.25
申请人 GLAXO GROUP LIMITED;ANDREWS, ROBERT, CARL;ANDERSEN, MARC, WERNER;STANFORD, JENNIFER, BADIANG;BUBACZ, DULCE, GARRIDO;CHAN, JOSEPH, HOWING;COWAN, DAVID, JOHN;GAUL, MICHAEL, DAVID;MCDOUGALD, DARRYL, LYNN;MUSSO, DAVID, LEE;RABINOWITZ, MICHAEL, HOWARD;WIETHE, ROBERT, WILLIAM 发明人 ANDREWS, ROBERT, CARL;ANDERSEN, MARC, WERNER;STANFORD, JENNIFER, BADIANG;BUBACZ, DULCE, GARRIDO;CHAN, JOSEPH, HOWING;COWAN, DAVID, JOHN;GAUL, MICHAEL, DAVID;MCDOUGALD, DARRYL, LYNN;MUSSO, DAVID, LEE;RABINOWITZ, MICHAEL, HOWARD;WIETHE, ROBERT, WILLIAM
分类号 C07D213/75;C07D277/46;C07D285/12;C07D285/135;C07D409/12;C07D417/12;(IPC1-7):A61K31/34;A61K31/35;A61K31/42;A61K31/44;A61K31/505;C07D211/04;C07D213/02;C07D239/02;C07D263/56;C07D307/79;C07D311/58;C07D319/20;C07D333/54 主分类号 C07D213/75
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