发明名称 |
2-OXO-2H-QUINOLINE DERIVATIVES |
摘要 |
The invention relates to novel compounds of formula (I), wherein X, Y, R, R1 , R2, R3 and n have the meaning cited in patent claim 1. Said compounds are inhibitors of coagulation factor Xa and can be used in the prophylaxis and/o r therapy of thromboembolic diseases.
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申请公布号 |
CA2342230(A1) |
申请公布日期 |
2000.03.09 |
申请号 |
CA19992342230 |
申请日期 |
1999.07.26 |
申请人 |
MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG |
发明人 |
MELZER, GUIDO;ANZALI, SOHEILA;BERNOTAT-DANIELOWSKI, SABINE;BUCHSTALLER, HANS-PETER;DORSCH, DIETER;MEDERSKI, WERNER;WURZIGER, HANNS;JURASZYK, HORST;GANTE, JOACHIM |
分类号 |
C07D215/22;A61K31/4704;A61K31/4709;A61P7/02;A61P9/10;A61P29/00;A61P43/00;C07D215/227;C07D215/50;C07D215/54;C07D413/10;C07D413/14;(IPC1-7):C07D215/22;C07D413/12;A61K31/47 |
主分类号 |
C07D215/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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