发明名称 |
Glycoprotein IIB IIIA antagonists |
摘要 |
This invention relates to certain bicyclic compounds having a nucleus formed of two fused six membered rings, for example, benzopyran, isoquinoline, isoquinolone, tetrahydronaphthalene, dihydronaphthalene, or tetralone, substituted with both basic and acidic functionality, which are useful in inhibition of platelet aggregation.
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申请公布号 |
US6020362(A) |
申请公布日期 |
2000.02.01 |
申请号 |
US19980047285 |
申请日期 |
1998.03.24 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
FISHER, MATTHEW J.;HAPP, ANNE MARIE;JAKUBOWSKI, JOSEPH A.;KINNICK, MICHAEL DEAN;KLINE, ALLEN D.;MARTINELLI, MICHAEL JOHN;MORIN, JR., JOHN MICHAEL;PAAL, MICHAEL;RUEHTER, GERD;RUTERBORIES, KENNETH JAMES;SALL, DANIEL J.;SCHOTTEN, THEO;SKELTON, MARSHALL A.;STENZEL, WOLFGANG;VASILEFF, ROBERT THEODORE |
分类号 |
C07D487/04;A61K31/195;A61K31/215;A61K31/335;A61K31/35;A61K31/352;A61K31/38;A61K31/381;A61K31/44;A61K31/4427;A61K31/443;A61K31/445;A61K31/4465;A61K31/47;A61K31/472;A61K31/495;A61P7/02;A61P9/10;C07C257/18;C07C257/20;C07C271/64;C07D211/22;C07D211/32;C07D211/34;C07D213/82;C07D217/04;C07D217/06;C07D217/24;C07D221/00;C07D311/22;C07D311/58;C07D311/66;C07D311/70;C07D319/16;C07D333/38;C07D401/12;C07D405/06;C07D405/12;C07D491/052;C07D497/04;G03F7/20;(IPC1-7):C07D311/04 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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地址 |
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