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发明名称
PROCESS FOR THE PREPARATION OF AN INDOLE DERIVATE
摘要
A process for the preparation of methyl 2-(3-chloropropoxy)-indole-3-carboxylate, which comprises reacting a 3-chloro-3-carboxylate indole compound with 3-chloropropanol in the presence of an acid having a pKa of from 0 to 2.
申请公布号
WO0003984(A1)
申请公布日期
2000.01.27
申请号
WO1999EP04944
申请日期
1999.07.13
申请人
SMITHKLINE BEECHAM PLC;FEDOULOFF, MICHAEL;STRACHAN, JOHN, BRYCE
发明人
FEDOULOFF, MICHAEL;STRACHAN, JOHN, BRYCE
分类号
C07D498/04;C07D209/42;(IPC1-7):C07D209/42
主分类号
C07D498/04
代理机构
代理人
主权项
地址
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