SYNTHESIS OF ARYL GLUCURONIDE OF 2-HYDROXY-N-(5-NITRO-2-THIAZOLYL) BENZAMIDE, AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME

摘要

An aryl glucuronide of 2-hydroxy-N-(5-nitro-2-thiazolyl)benzamide, preferably an O-aryl glucuronide, as well as methods for the convenient synthesis of these aryl glucuronides, highly stable and low toxicity pharmaceutical composition containing these aryl glucuronides, and methods for use of these pharmaceutical compositions, for example, for treatment of inflammation, infections, etc.