发明名称 FLUORINE-CONTAINING ALPHA-INDOLEPROPIONIC ACID COMPOUND, ITS PRODUCTION AND PLANT GROWTH REGULATOR WITH THE SAME AS ACTIVE INGREDIENT
摘要 PROBLEM TO BE SOLVED: To obtain the subject new compound having plant growth promotive activity. SOLUTION: This new compound is shown by formula I (Y is H or an alkyl; X<1> and X<2> are each H, an alkyl, alkoxy, aryl, or halogen), e.g. methyl 3,3,3- trifluoro-2-(indole-3-)propionate. The compound of formula I is obtained by the following procedure: a compound of formula II (R is H or an alkyl) is dissolved in a polar solvent such as dimethylformamide and then reacted with a chlorinating agent (e.g. thionyl chloride, oxalyl chloride) followed by reducing the reaction product with e.g. sodium borohydride and then, as necessary, carrying out hydrolysis under heating. When the compound of formula I is to be used as a plant growth regulator, it can be used either directly, or in the form of a preparation such as a liquid, powder, granules, wettable powder or flowable through mixing with an auxiliary commonly used in agrochemicals; it is preferable that the compound of formula I is used at a concentration of 1×10<-9> to 1×10<-2> M.
申请公布号 JPH11349569(A) 申请公布日期 1999.12.21
申请号 JP19980173941 申请日期 1998.06.04
申请人 AGENCY OF IND SCIENCE & TECHNOL 发明人 FUJII SHOZO;KATO KATSUYA;KATAYAMA MASATO;KIMOTO HIROSHI
分类号 C07D209/18;A01N43/38;C07D209/30;C07D209/34;(IPC1-7):C07D209/18 主分类号 C07D209/18
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