发明名称 HETEROCYCLIC CIS CYCLOPROPANE DERIVATIVES AS MELATONERGIC AGENTS
摘要 There is provided a novel series of cis cyclopropane compounds of Formula (I), wherein R<1>, R<2>, R<3>, R<4>, X, Y, Z and m are as defined herein which bind to the human melatonin receptor and therefore are useful as melatonergic agents.
申请公布号 WO9962515(A1) 申请公布日期 1999.12.09
申请号 WO1999US11474 申请日期 1999.05.25
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 CHEN, JIE;DEXTRAZE, PIERRE;DODIER, MARCO;TAKAKI, KATHERINE, S.
分类号 C07D307/81;A61K31/343;A61K31/36;A61P25/20;C07C233/05;C07D307/79;C07D317/48;(IPC1-7):A61K31/44;A61K31/335;A01N43/08;A01N43/30;A01N43/32;C07D307/88;C07D317/46;C07D319/04;C07D319/08 主分类号 C07D307/81
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