发明名称 |
HETEROCYCLIC CIS CYCLOPROPANE DERIVATIVES AS MELATONERGIC AGENTS |
摘要 |
There is provided a novel series of cis cyclopropane compounds of Formula (I), wherein R<1>, R<2>, R<3>, R<4>, X, Y, Z and m are as defined herein which bind to the human melatonin receptor and therefore are useful as melatonergic agents.
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申请公布号 |
WO9962515(A1) |
申请公布日期 |
1999.12.09 |
申请号 |
WO1999US11474 |
申请日期 |
1999.05.25 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
CHEN, JIE;DEXTRAZE, PIERRE;DODIER, MARCO;TAKAKI, KATHERINE, S. |
分类号 |
C07D307/81;A61K31/343;A61K31/36;A61P25/20;C07C233/05;C07D307/79;C07D317/48;(IPC1-7):A61K31/44;A61K31/335;A01N43/08;A01N43/30;A01N43/32;C07D307/88;C07D317/46;C07D319/04;C07D319/08 |
主分类号 |
C07D307/81 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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