发明名称 Substituted carbazoles, process for their preparation and their use as sPLA2 inhibitiors
摘要 <p>A class of novel tricyclics is disclosed together with the use of such compounds for inhibiting sPLA<Sub>2</Sub> mediated release of fatty acids for treatment of conditions such as septic shock.</p>
申请公布号 EP0952149(A2) 申请公布日期 1999.10.27
申请号 EP19990302941 申请日期 1999.04.16
申请人 ELI LILLY AND COMPANY 发明人 ANDERSON, BENJAMIN ALAN;BACH, NICHOLAS JAMES;BASTIAN, JOLIE ANNE;HARN, NANCY KAY;HARPER, RICHARD WALTZ;HITE, GARY ALAN;KINNICK, MICHAEL DEAN;LIN, HO-SHEN;LONCHARICH, RICHARD JAMES;MCGILL, JOHN MCNEILL;MIHELICH, EDWARD DAVID;MORIN JR., JOHN MICHAEL;PHILLIPS, MICHAEL LEROY;RICHETT, MICHAEL ENRICO;SALL, DANIEL JON;SAWYER,JASON SCOTT;SCHEVITZ, RICHARD WALTER;VASILEFF, ROBERT THEODORE
分类号 C07D401/06;A61K31/00;A61K31/40;A61K31/403;A61K31/44;A61K31/4427;A61K31/443;A61K31/4433;A61K31/4439;A61P1/00;A61P7/00;A61P11/00;A61P11/06;A61P19/00;A61P19/02;A61P29/00;A61P31/00;A61P31/04;A61P35/00;A61P43/00;C07C205/59;C07C229/48;C07C229/60;C07D209/82;C07D209/86;C07D209/88;C07D405/04;C07D409/04;(IPC1-7):C07D209/88 主分类号 C07D401/06
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