发明名称 USE OF SUBSTITUTED 2-MERCAPTONICOTINIC ACID DERIVATIVES FOR COMBATING ENDOPARASITES, NEW SUBSTITUTED 2-MERCAPTONICOTINIC ACID DERIVATIVES AND PROCESSES FOR THEIR PREPARATION
摘要 Use of substituted 2-mercaptonicotinic acid derivatives for combating endoparasites, new substituted 2-mercaptonicotinic acid derivatives and processes for their preparation The present invention relates to the use of compounds of the general formula I I in which R1 represents C1-C8-alkyl, aralkyl, aryl or heteroaryl radicals which are optionally substituted by halogen, cyano, nitro, amino, alkylamino, aminoacyl, alkyl, aralkyl, halogenoalkyl, alkoxy, aryloxy, halogenoalkoxy, alkylthio, arylthio, alkylsulphinyl, arylsulphinyl, arylsulphonyl, halogenoalkylthio, haloganoalkylsulphinyl, halogenoalkylsulphonyl or carbonylaryl, X represents O, or / N-R3, R2 represents C1-5-alkyl, aralkyl, alkenyl or alkinyl, R3 represents H or alkyl or R1 and R3, together with the adjacent N atom, represent a 5 or 6-membered heterocycle which can contain O or N as additional heteroatoms and is optionally substituted by C1-4-alkyl, Le A 27 948 R4 represents hydrogen, halogen, alkyl, halogenoalkyl, cyano, nitro, amino, aminoacyl, phenyl, alkoxy, aryloxy, thioalkyl and arylthio which are optionally substituted, for combating endoparasites in medicine and veterinary medicine. Le A 27 9413
申请公布号 CA2052894(A1) 申请公布日期 1992.04.11
申请号 CA19912052894 申请日期 1991.10.07
申请人 BAYER AKTIENGESELLSCHAFT 发明人 BONSE, GERHARD;JESCHKE, PETER;LINDNER, WERNER;HARDER, ACHIM;MENCKE, NORBERT
分类号 A61K31/455;A61K31/4418;A61K31/4427;A61P33/10;C07D213/80;C07D213/82;C07D401/12;(IPC1-7):C07D213/82;C07D407/12;C07D409/12;C07D413/12;C07D417/12;A01N43/40;A61K31/44;A61K31/535;C07D213/84 主分类号 A61K31/455
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