发明名称 |
4-AMINO-(ETHYLAMINO)-OXINDOLE DOPAMINE AUTORECEPTOR AGONISTS |
摘要 |
Compounds having dopaminegic activity are provided, having formula (I) wherein R<1> and R<2> are each, independently, hydrogen, C1-10 alkyl, or (CH2)mR<4>, wherein R<4> is phenyl or naphthyl which may be substituted by one or two substituents selected from the group consisting of C1-6 alkyl, halogen, C1-6 alkoxide and trifluoromethyl and m is 1 to 5; and R<3> is hydrogen or C1-6 alkyl; or pharmaceutically acceptable salts thereof.
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申请公布号 |
WO9952870(A1) |
申请公布日期 |
1999.10.21 |
申请号 |
WO1999US07967 |
申请日期 |
1999.04.12 |
申请人 |
AMERICAN HOME PRODUCTS CORPORATION |
发明人 |
NELSON, JAMES, ALBERT;KANZELBERGER, MIRA, ANA;MEWSHAW, RICHARD, ERIC |
分类号 |
A61K31/404;A61K31/403;A61P25/00;A61P25/16;A61P25/18;A61P25/30;A61P43/00;C07D209/34;(IPC1-7):C07D209/34;A61K31/40 |
主分类号 |
A61K31/404 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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