发明名称 Piperidine derivatives.
摘要 Piperidine derivatives of the formula Iand their physiologically acceptable saltsin which X, Y, Z, R1, R2, R3 and R4 are as defined in claim 1can be as excitatory amino acid antagonists for combating neurodegenerative disorders including cerebrovascular diseases, epilepsy, schizophrenia, Alzheimer's disease, Parkinson's disease and Huntington's disease, cerebral ischaemias, infarcts and psychosis.
申请公布号 ZA9902191(B) 申请公布日期 1999.09.29
申请号 ZA19990002191 申请日期 1999.03.18
申请人 MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG 发明人 HELMUT PRUECHER;ANDREW BARBER;JOACHIM LEIBROCK;GERD BARTOSZYK
分类号 A61K31/4427;A61K31/445;A61K31/454;A61K31/4709;A61P9/10;A61P25/00;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/28;A61P43/00;C07D401/06;C07D413/06;C07D417/06 主分类号 A61K31/4427
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