发明名称 |
Processes for the preparation of (r)-alpha- (2,3-dimethoxyphenyl)- 1-Ý2-(4- fluorophenyl)ethyl¨- 4-piperidinemethanol |
摘要 |
The present invention provides various processes for the preparation of (R)-±-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol. These processes may be characterized by the following scheme: |
申请公布号 |
AU2998899(A) |
申请公布日期 |
1999.09.27 |
申请号 |
AU19990029988 |
申请日期 |
1999.03.11 |
申请人 |
HOECHST MARION ROUSSEL, INC.;HOECHST MARION ROUSSEL DEUTSCHLAND GMBH |
发明人 |
ALAN G. BINA;EDWARD D. DAUGS;JONATHAN C. EVANS;HANS-WOLFRAM FLEMMING;GERARD GUILLAMOT;ROBERT A. HAWTHORNE;THOMAS H. E. HILPERT;JAMES E. HITT;CHI-HSIN R. KING;JOHANNES N. KOEK;FREDERICK M. LASKOVICS;JOHN R LEFLER;ALEXEY L. MARGOLIN;SHARON K MINISH;THOMAS T ORTYL;LIAN G. RAJEWSKI;MARVIN J. SACK;PAUL F. SKULTETY |
分类号 |
A61K9/20;A61K31/4409;A61K31/445;A61K47/04;A61K47/12;A61K47/26;A61K47/38;A61P1/14;A61P7/02;A61P9/06;A61P9/08;A61P9/10;A61P21/00;A61P25/00;A61P25/18;A61P25/22;C07D211/22;C07D211/32;C07D213/00;C07D213/50 |
主分类号 |
A61K9/20 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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