发明名称 SYNTHESIS OF EPOTHILONES, INTERMEDIATES THERETO AND ANALOGUES THEREOF
摘要 The present invention provides convergent processes for preparing epothilone A and B, desoxyepothilones A and B, and analogues thereof, useful in the treatment of cancer and cancer which has developed a multidrug-resistant phenotype. Also provided are intermediates useful for preparing said epothilones.
申请公布号 CA2322157(A1) 申请公布日期 1999.09.02
申请号 CA19992322157 申请日期 1999.02.24
申请人 SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH 发明人 DANISHEFSKY, SAMUEL J.;BALOG, AARON;BERTINATO, PETER;SORENSEN, ERIK J.;KUDUK, SCOTT;KAMENECKA, TED;CHOU, TING-CHAU;MENG, DONGFANG;BERTINO, JOSEPH R.;ZHANG, XIU-GUO;HARRIS, CHRISTINA;SU, DAI-SHI;SAVIN, KENNETH A.
分类号 A61K31/365;A61K31/427;A61P35/00;C07C59/185;C07C59/76;C07C69/66;C07C69/738;C07D233/54;C07D277/24;C07D277/28;C07D277/30;C07D313/00;C07D417/06;C07D493/04;C07F7/02;C07F7/18;(IPC1-7):C07D209/12;C07D277/08;C07D277/22;A61K31/335;C07D263/34;A61K31/415;A61K31/42;A61K31/425;A61K31/44 主分类号 A61K31/365
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