发明名称 |
N-[2-substituted-3-(2-aminoethyl)-1H-indol-5-YL]-Amides: new 5-HT1F agonists |
摘要 |
PCT No. PCT/US96/16122 Sec. 371 Date Mar. 13, 1998 Sec. 102(e) Date Mar. 13, 1998 PCT Filed Oct. 8, 1996 PCT Pub. No. WO97/13512 PCT Pub. Date Apr. 17, 1997The invention provides novel 5-HT1f agonists of formula (I) where X, R1, R2, and R3 are defined in the specification, which are useful for the treatment of migraine and associate disorders.
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申请公布号 |
US5942536(A) |
申请公布日期 |
1999.08.24 |
申请号 |
US19980043360 |
申请日期 |
1998.03.13 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
FRITZ, JAMES E;HAHN, PATRIC J;KALDOR, STEPHEN W;SIEGEL, MILES G;XU, YAO-CHANG |
分类号 |
C07D401/04;A61K31/00;A61K31/40;A61K31/403;A61K31/404;A61K31/4045;A61K31/415;A61K31/4155;A61K31/42;A61K31/44;A61K31/4427;A61K31/443;A61K31/4433;A61K31/4439;A61K31/47;A61K31/472;A61K31/4725;A61K31/495;A61K31/498;A61K31/74;A61P25/00;A61P43/00;C07D209/14;C07D209/16;C07D401/12;C07D403/04;C07D403/12;C07D405/12;C07D409/04;C07D409/12;C07D413/12;C07D417/12;(IPC1-7):A61K31/405;C07D209/08 |
主分类号 |
C07D401/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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