发明名称 ACETAMIDO-2,3,4,5-TETRADIOXY-4-GYANIDINO-D-GLYCERO-D- GALACTONONE-2-ENOPYRANOZONIC ACID IN CRYSTALLINE FORM, PREPARATION METHODS, PHARMACEUTICAL COMPOSITION, AND METHOD OF PREPARING THEREOF
摘要 FIELD: pharmaceutical industry. SUBSTANCE: described are particular physical forms of 5-acetamido-2,3,4,5-tetradeoxy-4-guanidino-3- glycero-D-galactonone-2-enopyranozonic acid, more particularly in crystalline form in which all crystalline water is substantially lost at 80-90 C, 5-acetamido, 2,3,4,5-tetradeoxy-4-guanidino-D-glycero-D-galactonone-2- enopyranozonic acid is included into pharmaceutical composition for use as antiviral agent. EFFECT: improved properties of the pharmaceutical composition. 33 cl, 1 dwg, 11 ex, 2 tbl
申请公布号 RU2134690(C1) 申请公布日期 1999.08.20
申请号 RU19960115122 申请日期 1994.12.15
申请人 BIOTA SAJENTIFIK MENEDZHMENT PTI LTD. 发明人 KRISTOFER VIL'JAMSON;VIL'JAM DZHEJMS VAJT;VIPULKUMAR PATEL
分类号 A61K31/35;A61K31/351;A61P31/12;C07D309/28;(IPC1-7):C07D309/28 主分类号 A61K31/35
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