发明名称 |
NOVEL CYCLIC SULFONAMIDE DERIVATIVES AS METALLOPROTEINASE INHIBITORS |
摘要 |
The present application describes novel lactams and derivatives thereof of formula (I) or pharmaceutically acceptable salt forms thereof, wherein ring B is a 4-8 membered cyclic sulfonamide containing from 0-3 additional heteroatoms selected from N, O, and S, which are useful as metalloprotease inhibitors.
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申请公布号 |
WO9941246(A1) |
申请公布日期 |
1999.08.19 |
申请号 |
WO1999US02767 |
申请日期 |
1999.02.10 |
申请人 |
DU PONT PHARMACEUTICALS COMPANY |
发明人 |
DUAN, JINGWU;CHEN, LIHUA;CHERNEY, ROBERT, J.;DECICCO, CARL, P.;VOSS, MATTHEW, E. |
分类号 |
A61K31/5415;A61K31/554;A61P1/02;A61P7/02;A61P7/04;A61P9/14;A61P17/06;A61P19/02;A61P25/00;A61P25/32;A61P27/02;A61P27/06;A61P29/00;A61P31/00;A61P31/18;A61P35/00;A61P35/04;A61P37/02;A61P43/00;C07D279/02;C07D285/36;C07D417/06;C07D417/12;(IPC1-7):C07D285/36;A61K31/55;A61K31/54 |
主分类号 |
A61K31/5415 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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