发明名称 BIARYL-ACETIC ACID DERIVATIVES AND THEIR USE AS COX-2 INHIBITORS
摘要 The present invention relates to inhibitors of COX-2, compositions which contain such compounds and methods of use. The compounds are represented by formula (I) and include pharmaceutically acceptable salts and esters thereof.
申请公布号 WO9941224(A1) 申请公布日期 1999.08.19
申请号 WO1999CA00120 申请日期 1999.02.11
申请人 MERCK FROSST CANADA & CO.;BAYLY, CHRISTOPHER, I.;BLACK, CAMERON;OUIMET, NATHALIE;PERCIVAL, DAVID;LEGER, SERGE;OUELLET, MARC 发明人 BAYLY, CHRISTOPHER, I.;BLACK, CAMERON;OUIMET, NATHALIE;PERCIVAL, DAVID;LEGER, SERGE;OUELLET, MARC
分类号 C07D333/60;A61K31/192;A61K31/216;A61K31/34;A61K31/343;A61K31/381;A61K31/403;A61K31/4035;A61K31/404;A61K31/41;A61K31/4184;A61K31/423;A61K31/428;A61K31/437;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/495;A61K31/496;A61K31/4985;A61P1/00;A61P3/10;A61P11/06;A61P15/06;A61P19/02;A61P19/06;A61P19/10;A61P25/04;A61P25/06;A61P25/28;A61P27/02;A61P27/06;A61P29/00;A61P31/12;A61P35/00;A61P35/04;A61P37/02;A61P43/00;C07C57/42;C07C59/64;C07C69/618;C07C69/734;C07C323/62;C07D209/08;C07D209/18;C07D209/44;C07D213/55;C07D213/64;C07D213/69;C07D235/08;C07D263/56;C07D277/64;C07D307/79;C07D333/54;C07D471/04;(IPC1-7):C07C59/64;A61K31/19;A61K31/215;A61K31/40;A61K31/38 主分类号 C07D333/60
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