发明名称 ANTIMYCOTICALLY ACTIVE CYCLOPROPYL-SUBSTITUTED AZOLYLMETHYLCARBINOLS
摘要 Antimycotically active 1-cyano- and 1-carboxamidocyclopropylazolylmethylcarbinols have now been found of the formula (see fig. I) in which R1 - represents hydrogen or - represents alkyl or - represents alkylcarbonyl, R2 - represents cyano or - represents a group of the formula (see fig. II) R3 - represents phenyl which is optionally substituted by halogen, straight-chain or branched alkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy or halo-genoalkylthio, or by phenyl or phenoxy which, in turn, may be substituted by halogen or alkyl having up to 6 carbon atoms, X - represents a nitrogen atom or the CH group, Y - represents a bond or - represents a group of the formula (see fig. III, IV) or -C~C-in which R4 and R5 are identical or different and denote hydrogen or alkyl and their pharmaceutically tolerated acid addition salts.
申请公布号 CA2003213(C) 申请公布日期 1999.08.03
申请号 CA19892003213 申请日期 1989.11.17
申请人 发明人 STROECH, KLAUS;BUECHEL, KARL HEINZ;FUGMANN, BURKHARD;PLEMPEL, MANFRED
分类号 A01N53/12;A61K31/41;A61K31/415;A61P31/04;C07C255/45;C07C255/46;C07C323/20;C07C323/62;C07D233/60;C07D233/61;C07D249/08;C07D521/00;(IPC1-7):C07D233/61 主分类号 A01N53/12
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