| 发明名称 |
BISULFATE SALT OF HIV PROTEASE INHIBITOR |
| 摘要 |
The present invention provides the crystalline bisulfate salt of formula (II) which is found to have unexpectedly high solubility/dissolution rate and oral bioavailability relative to the free base form of this azapeptide HIV protease inhibitor compound.
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| 申请公布号 |
WO9936404(A1) |
申请公布日期 |
1999.07.22 |
| 申请号 |
WO1998US27382 |
申请日期 |
1998.12.22 |
| 申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
SINGH, JANAK;PUDIPEDDI, MADHUSUDHAN;LINDRUD, MARK, D. |
| 分类号 |
C07K5/02;A61K31/44;A61K31/4402;A61K31/4418;A61K38/05;A61P31/18;A61P43/00;C07D213/02;C07D213/42;(IPC1-7):C07D213/02 |
主分类号 |
C07K5/02 |
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